Laroprovstat + Ezetimibe Bioavailability Study

AC
Overseen ByAstraZeneca Clinical Study Information Center
No Placebo GroupAll trial participants will receive the active study treatment (no placebo)

What You Need to Know Before You Apply

What is the purpose of this trial?

The purpose of this study is to assess how well laroprovstat and ezetimibe combined in a single tablet to be taken by mouth works and what the body does to the drug (pharmacokinetics) compared with laroprovstat and ezetimibe individual tablets to be taken by mouth (relative bioavailability) as well as to see if there is any effect of eating compared to fasting (food effect) in healthy adults.

Are You a Good Fit for This Trial?

This trial is for healthy adults. People with certain health conditions, like high cholesterol or diabetic dyslipidemia, may be of interest in future studies, but only those without significant medical issues can join this phase.

Inclusion Criteria

Have a Body mass index (BMI) between 18 and 30 kg/m2 inclusive and weigh at least 50 kg
I am a healthy adult between 18 and 55 years old.
I am female and have tested negative for pregnancy before starting the study.
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Exclusion Criteria

History of severe allergy/hypersensitivity or ongoing clinically important allergy/hypersensitivity to drugs with a similar chemical structure or class to laroprovstat or ezetimibe
I have not taken PCSK9 inhibitors in the past year or inclisiran ever.
History of any clinically important disease or disorder
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Timeline for a Trial Participant

Screening

Participants are screened for eligibility to participate in the trial

2-4 weeks

Treatment

Participants receive single-dose treatments in a randomized, open-label, 4-period, cross-over design to assess the relative bioavailability of laroprovstat/ezetimibe fixed combination drug products versus single therapy products.

44 days
4 treatment periods, each lasting 11 days

Washout

Washout periods between treatment phases to clear the drug from the body before the next treatment period begins.

Variable

Follow-up

Participants are monitored for safety and effectiveness after treatment

4 weeks

What Are the Treatments Tested in This Trial?

Trial Overview

The study compares how the body absorbs and processes a combined tablet of laroprovstat and ezetimibe versus taking each drug separately. It also looks at whether eating affects how these drugs work. Participants receive all treatments at different times.

How Is the Trial Designed?

4

Treatment groups

Experimental Treatment

Group I: Treatment DExperimental Treatment1 Intervention
Group II: Treatment CExperimental Treatment1 Intervention
Group III: Treatment BExperimental Treatment2 Interventions
Group IV: Treatment AExperimental Treatment1 Intervention

Find a Clinic Near You

Who Is Running the Clinical Trial?

AstraZeneca

Lead Sponsor

Trials
4,491
Recruited
290,540,000+

Sir Pascal Soriot

AstraZeneca

Chief Executive Officer since 2012

Veterinary Medicine from École nationale vétérinaire d'Alfort, MBA from HEC Paris

Dr. Cristian Massacesi

AstraZeneca

Chief Medical Officer since 2021

MD from Marche Polytechnic University, Oncology training at Royal Marsden Hospital, Kaplan Comprehensive Cancer Center, and European Institute of Oncology

Pascal Soriot

AstraZeneca

Chief Executive Officer since 2012

Veterinary Medicine from École nationale vétérinaire d'Alfort, MBA from HEC Paris

Cristian Massacesi

AstraZeneca

Chief Medical Officer since 2021

MD from Marche Polytechnic University, Medical Oncology training at Royal Marsden Hospital, Kaplan Comprehensive Cancer Center, and European Institute of Oncology